平安! 发表于 2011-11-9 19:57
# B: b9 z0 \. n, u: L# U% i KPazopanib (100 mg/kg/day free base equivalent)
" A% @' a- i$ D0 {; |( w$ v8 u5 w8 l 这是个已经在美国上市的老药了,能下载到正式药物使用说明书英文版。
5 ?9 ^6 T$ ` d* |* h搜索了一下,原料一大堆。
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对不起!100mg/kg是用于移植瘤的,我弄错了。
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以下是正版说明书的推荐用量。7 E5 K& P% `+ {6 P: s& B# r. Y
! L0 f% T3 m* r3 l! p- u--------------------- DOSAGE AND ADMINISTRATION ----------------
: }* C) F$ u* r5 i1 }5 m# k8 r; D* 800 mg orally once daily without food (at least 1 hour before or 2 hours after a meal). (2.1) 2 t5 T2 U+ y" ?) y/ @
* Baseline moderate hepatic impairment – 200 mg orally once daily. Not recommended in patients with severe hepatic impairment. (2.2) 6 ]2 V7 B; \& c
---------------------DOSAGE FORMS AND STRENGTHS --------------
7 [: d: `) ]( v n+ u; g- s+ P200 mg tablets. (3)
! H. o6 C; f1 {- w6 H( S) {-------------------------------CONTRAINDICATIONS------------------------ |