平安! 发表于 2011-11-9 19:57 3 L* c8 h, U i$ h8 t( H
Pazopanib (100 mg/kg/day free base equivalent) & T; f2 Y2 w: B7 w+ z$ L9 Y
这是个已经在美国上市的老药了,能下载到正式药物使用说明书英文版。4 U+ `6 n* t8 n8 i, v( r2 h
搜索了一下,原料一大堆。& e! t' d1 c- m
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对不起!100mg/kg是用于移植瘤的,我弄错了。
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. `# x3 y( r" l! E+ \; A以下是正版说明书的推荐用量。: b+ O7 X+ d0 I- w0 r, _' h$ {
6 N, \2 ^1 J/ l3 s--------------------- DOSAGE AND ADMINISTRATION ----------------) {6 K9 _9 K7 G' c- E
* 800 mg orally once daily without food (at least 1 hour before or 2 hours after a meal). (2.1)
" E: f% Y0 a" ~5 p/ w5 [. J* Baseline moderate hepatic impairment – 200 mg orally once daily. Not recommended in patients with severe hepatic impairment. (2.2) ' U3 ]0 \4 V' | [+ ?# l
---------------------DOSAGE FORMS AND STRENGTHS --------------2 S) J, q6 I( n' h8 J7 P
200 mg tablets. (3) ) H" Z( u( t- ?' `
-------------------------------CONTRAINDICATIONS------------------------ |